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CMP-5

Glpbio
Catalog No:GC39665-10mM (in 1mL DMSO) CAS No.:880813-42-3 MDLNo: Brand:Glpbio purity: 特性: Purpose:CMP-5 是一種有效的選擇性 PRMT5 抑制劑,對 PRMT1,PRMT4 和 PRMT7 酶無活性。CMP-5 在組蛋白的準備過程中,通過抑制 PRMT5 甲基轉移酶活性選擇性地阻斷 S2Me-H4R3。CMP-5 阻斷 EBV 驅動的 B 淋巴細胞轉化,但對正常 B 細胞沒有影響。DMSO: 125 mg/mL (396.31 mM)
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